Efficient and divergent synthesis of cyclophosphamide analogues from 2-arylamino-3-acetyl-5,6-dihydro-4H-pyrans.

نویسندگان

  • Dexuan Xiang
  • Peng Huang
  • Kewei Wang
  • Guangyuan Zhou
  • Yongjiu Liang
  • Dewen Dong
چکیده

A facile and efficient one-pot synthesis of substituted cyclophosphamidic chlorides and their analogues has been developed from readily available enaminones, 2-arylamino-3-acetyl-5,6-dihydro-4H-pyrans.

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عنوان ژورنال:
  • Chemical communications

دوره 46  شماره 

صفحات  -

تاریخ انتشار 2008